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Peptide Drug Interactions Database

A comprehensive reference for clinical peptide-drug interactions.

SeverityMeaning
MajorAvoid combination; significant risk
ModerateUse with caution; monitor closely
MinorLow risk; monitor
PeptideInteracting DrugSeverityEffectRecommendation
SemaglutideInsulinModerateIncreased hypoglycemia riskReduce insulin dose
SemaglutideOral contraceptivesMinorDelayed absorptionUse barrier method
SemaglutideWarfarinMinorMonitor INRCheck INR regularly
LiraglutideInsulinModerateIncreased hypoglycemiaDose adjustment
ExenatideMetforminMinorGI effectsTake with food
DulaglutideInsulinModerateHypoglycemia riskReduce insulin
PeptideInteracting DrugSeverityEffectRecommendation
CJC-1295InsulinModerateHypoglycemiaMonitor glucose
IpamorelinCorticosteroidsMinorBlunted GH responseMonitor IGF-1
GHRP-6Dopamine agonistsMinorEnhanced GH releaseMonitor levels
TesamorelinInsulinModerateGlucose alterationAdjust insulin
PeptideInteracting DrugSeverityEffectRecommendation
OxytocinErgot alkaloidsMajorHypertension riskAvoid combination
DesmopressinLithiumModerateWater intoxicationMonitor sodium
DesmopressinNSAIDsMinorIncreased effectMonitor
PeptideInteracting DrugSeverityEffectRecommendation
BPC-157NSAIDsMinorEnhanced GI healingSafe combination
BPC-157AntihypertensivesMinorBP loweringMonitor
TB-500CorticosteroidsMinorEnhanced tissue repairSafe combination
GHK-CuTetracyclinesMinorChelation possibleSeparate dosing
  1. Monitor glucose with all GH/GLP-1 peptides + insulin
  2. Avoid ergot alkaloids with oxytocin
  3. Separate dosing for chelating peptides (GHK-Cu) + antibiotics
  4. Check INR with anticoagulants + GLP-1 RAs
  5. Monitor electrolytes with desmopressin + lithium